Thursday, June 23, 2016

Cardiac cachexia: A systematic overview

INTRODUCTION
- The incidence of CHF in the European and the United States is about 0.1-0.5% per ear; while the prevalence of CHF is about 0.3-2.4% (~5 million people) in the United States.
- About half of the patients with chronic heart failure (CHF) die within 4 years of diagnosis
- In unselected patients with CHF, mortality rates were as high as 50% in the cachectic subset compared to 17% in the non-cachectic subset at 18 months of follow-up.
- Cachexia is not only associated with poor outcomes, but also with an unfavourable response to drug treatment and poor quality of life

DEFINITION OF CARDIAC CACHEXIA
- Cardiac cachexia as a clinical entity is acknowledged as a complex syndrome, which is associated with poor outcomes.
- No single reason for cachexia exists
- Patients usually experience progressive weight loss with body composition alterations and disturbed homeostasis of several body systems.
- There is evidence for activation of neuroendocrine and inflammatory systems, increased lipolysis, muscle wasting, lack of appetite, and malabsorption whilst the importance of individual pathways and the exact interplay remain unknown.
-The authors proposed definition: non-oedematous weight loss of >6% of total body weight over a period of 6 or more months (At this stage it is important to note that the severity of cardiac cachexia may not always correlate with classical criteria of disease severity as New York Heart Association [NYHA] functional class, left ventricular ejection fraction, or exercise duration; Cardiac cachexia even may not be associated with morphological cardiac changes as seen by magnetic resonance imaging or echocardiography)
- It might be necessary to add some laboratory, clinical and functional parameters to be able to identify cachexia and body wasting in an early phase.
- Ideally, patients at risk for the development of cachexia should be identified as early as possible, however, no effective treatment of manifest cachexia is available yet.
- The definition by Evans 2008 may also be relevant.

Cautious with terms such as “cachexia”, “anorexia”, “sarcopenia”, “malnutrition” and “hypercatabolism” – they are not the same!
- Sarcopenia: age associated “normal” muscle wasting, may not result in significant weight changes, because loss of muscle and increases in fat mass are frequently balanced.
- Malnutrition and Anorexia: are associated with predominantly loss of fat mass rather than muscle tissue; are reversible with adequate food intake, but not cachexia
- Hypercatabolism cannot be evaluated during clinical examination and neglects the other side of the coin, the anabolic processes

PATHOPHYSIOLOGICAL ASPECTS OF CARDIAC CACHEXIA
1) Immune Activation
- One key aspect of CHF and cardiac cachexia like many other forms of cachexia is inflammatory immune activation
- Activation of the pro-inflammatory mediator tumour necrosis factor-α (TNFα) is the final common pathway that links all forms of cachexia.
- One of the most important signal transducers of many inflammatory stimuli is nuclear factor-κB (NF-κB).
- Interestingly, over-activity of the NF-κB system has been shown to occur in patients with CHF

2) Regulation of Feeding
- Feeding is a key component of a satiety-hunger homeostaticmodel (Fig.1).
- Although a simple but vital daily process, it is influenced by many pathways and/or mechanisms, which are still not completely understood (Table 2)
- The hypothalamus has been identified as the central regulating site of appetite (Fig. 2).
- Two areas can be differentiated: a lateral “feeding area” and a medial “satiety centre”
- Excessive fluctuations in feeding cause weight and body composition changes which may develop into medical conditions or disease
- Cachexia of chronic illnesses shares several nutritional features.
- Especially patients with cardiac cachexia experience appetite problems and alterations in food intake, malabsorption of nutrients, metabolic disturbances, and finally an anabolic/catabolic imbalance
- Malnourishment due to lack of appetite can occur in a variety of chronic diseases and as many as half of the patients can be affected.
- Disturbances in energy expenditure can contribute to anorexia-mediated body wasting and eventually to cachexia.
- Therefore, it is a key element in treating chronic illnesses that such patients receive adequate nutrition in order to prevent further development of the disease, to avoid potential side effects of treatment, and to recover from a state of deterioration.

3) Mechanisms of wasting in different body compartments
a)  Skeletal muscle is lost due to an imbalance of protein synthesis and proteolysis
- Typically proinflammatory cytokines induce proteolytic systems, while simultaneously reducing the anabolic IGF-1 signalling.
- Additionally myostatin, a negative regulator of muscle mass, is considered to be a key player, as it has been reported as up-regulated in HIV cachexia and sarcopenia

b) Later in the course of the disease, wasting of bone and fat mass is found
- Fat wasting can be induced by numerous agents and the rate limiting step is the activity of the enzyme hormone sensitivity lipase that can be activated by several receptors including β-adrenergic and natriuretic peptides receptors.
- TNFα, which is also over-expressed in both CHF and cardiac cachexia, plays a major role in fat cell lipolysis and inhibiting insulin signalling. The latter is an important aspect in the development of insulin resistance.
- It is tempting to speculate that increased levels of catecholamines and possibly natriuretic peptides may be responsible for the loss of adipose tissue that has been observed in such patients
- The bone density in patients with cardiac cachexia is lower, and lower calcium and vitamin D levels have been reported, although no mechanisms have been identified so far

- These alterations in body composition have their reasons in profound metabolic perturbations, which are initially meant to isolate and neutralize the insult that caused the heart to fail.
- However, at a later stage, they contribute to the development and the progression of cardiac cachexia.

THERAPEUTIC APPROACHES TO CARDIAC CACHEXIA
- Currently there are no approved therapies to treat of weight loss as such in cardiac cachexia

1) Prevention of Weight Loss
a) ACE Inhibitors & Beta-blockers
- Angiotensin Converting Enzyme (ACE) inhibitors and beta-blockers have both clinically shown their potential to delay and possibly prevent the onset of cardiac cachexia.

2) Nutrition
a) Feeding
- Although feeding alone, the reversal of the clinically observed anorexia, does not reverse cachexia, nutrition itself still seems to be a major factor in treatment strategies
- Often patients have deficiencies in micronutrients such as vitamins and a supplementation of branched-chain amino acids has shown to be beneficial
- An overall induction of food intake to battle anorexia in these patients is considered supportive.

b) Nutritional Consideration
- However, the daily sodium intake should be restricted to 2 g in all patients with advanced CHF or cardiac cachexia
- Prolonged periods of fasting are potentially harmful, and cachectic patients should be advised to eat small, frequent meals
- Fluid intake should be restricted to 1.5–2.0 l/day, especially in patients with severe symptoms or those requiring high doses of diuretics
- At least one study suggests that multiple micronutrient supplementation is potentially beneficial. Such supplements should contain anti-oxidant supplements and B-group vitamins
- Avoid food and lifestyle factors that trigger the acute phase response such as an excess of carbohydrates or saturated fats, alcohol, and smoking
- Food that counteracts inflammatory responses, can be recommended. This includes fish oil supplements, olives, walnuts, flaxseed oil, any fruits or vegetables, garlic, ginger, turmeric, sunflower seeds, eggs, herring, or nuts
- Enteral nutrition should always be given preference over parenteral nutrition, however, if the latter cannot be avoided, the general guidelines can be followed: 35 kcal per kg of bodyweight per day,1.2 g of protein per kg per day, and a 70:30 glucose:lipid ratio for the non-protein energy (ZYL note: I recommend to start slow while monitor for refeeding syndrome; increase calorie intake slowly as tolerated and prevent overfeeding)

3) Pharmacotherapy

I) Appetite Stimulants
a) Megestrol Acetate
- Megestrol acetate has been shown to stop weight loss in hormone responsive cancer and has recently been approved for AIDS cachexia in the United States.
- The closely related compound, medroxyprogesterone acetate, has similar effects, but a trend towards peripheral oedema was observed. Cannabinoids

b) Cannabinoids
- Cannabinoids are known inducers of food intake, but have clinically shown contradictory results.
- While positive effects on appetite were seen in patients with AIDS and cancer, there was no concomitant weight gain.

II) Anabolic agent
a) Anabolic Steroids
- The use of anabolic steroids in cachexia patients is limited to chronic obstructive pulmonary disease and AIDS, where positive effects on weight have been observed
- In CHF, there was an improved cardiac function, but no effect on weight

b) Beta-adrenergic agonist
- Beta-adrenergic, especially β2-adrenergic agonists are also known for their anabolic properties and have shown some beneficial effects in degenerative muscle diseases.
- Although short-lived, positive cardiac effects have been reported in CHF, but there was no improvement in the functional capacity of the patients

III) Anti-inflammatory strategies
- a) Neutralizing antibodies like eternacept and infliximab, which showed a lack of efficiency in CHF,
- b) Statins, which show beneficial pleiotropic effects like the reduction of pro-inflammatory cytokines in some settings and
- c) Thalidomide, which potently reduces TNFα

IV) Inhibition of major proteolysis pathway
- The use of proteasome inhibitors to inhibit major proteolysis pathway, the ubiquitin-proteasome pathway is in its early stages and has so far only been tested in cancer, where weight gain has been reported.
- While pentoxifylline reduced the activity of muscle proteolytic systems in a rat model of cancer cachexia, it failed to improve weight in patients with cancer cachexia.

CONCLUSION
- The pathophysiology of cardiac cachexia is exceedingly complex, and we still do not understand when and how CHF progresses into this syndrome
- Pro-inflammatory cytokines and especially TNFα certainly play an important part. However, therapies that targeted specific single cytokines have largely failed, and it appears that broader approaches are required.
- We are currently not able to interfere with appetite regulation in a promising way, although initial steps have been undertaken.
- Nutritional recommendations for cardiac cachexia remain speculative, and no large-scale randomized, controlled trials have been performed

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